← Pipeline|Gozebrutinib

Gozebrutinib

Approved
TEM-6828
Source: Trial-derived·Trials: 4
Modality
Peptide
MOA
BCL-2i
Target
Tau
Pathway
Innate Imm
CRCWilms
Development Pipeline
Preclinical
~Oct 2009
~Jan 2011
Phase 1
~Apr 2011
~Jul 2012
Phase 2
~Oct 2012
~Jan 2014
Phase 3
~Apr 2014
~Jul 2015
NDA/BLA
~Oct 2015
~Jan 2017
Approved
Apr 2017
Jul 2030
ApprovedCurrent
NCT03326700
1,011 pts·CRC
2024-092028-04·Completed
NCT07488696
1,680 pts·Wilms
2017-042026-10·Active
NCT05693685
2,531 pts·CRC
2023-022028-02·Terminated
+1 more trial
6,449 total pts2 indications
CompletedCurrentUpcoming
Catalysts (4)
2026-10-146mo awayPh3 Readout· Wilms
2028-02-171.9y awayPh3 Readout· CRC
2028-04-192.1y awayPh3 Readout· CRC
2030-07-034.3y awayPh3 Readout· CRC
Trial Timeline
2017Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
Approved
Active
Approved
Recruit…
Approved
Termina…
Approved
Complet…
Catalysts
Ph3 Readout
2026-10-14 · 6mo away
Wilms
Ph3 Readout
2028-02-17 · 1.9y away
CRC
Ph3 Readout
2028-04-19 · 2.1y away
CRC
Ph3 Readout
2030-07-03 · 4.3y away
CRC
RecruitingActiveCompletedTerminated|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT03326700ApprovedCRCCompleted1011VA
NCT07488696ApprovedWilmsActive1680BodyWt
NCT05693685ApprovedCRCTerminated2531BodyWt
NCT05777556ApprovedCRCRecruiting1227MRD
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-5501PfizerPhase 1BTKBCL-2i
RHH-3592RochePhase 1/2GIP-RBCL-2i
GeliderotideNovartisNDA/BLAIL-17ABCL-2i
NVO-9087Novo NordiskPhase 1/2TauCAR-T BCMA
TezecilimabTakedaNDA/BLATauBCL-2i
TAK-8262TakedaNDA/BLATauTNFi
RimaosocimabAmgenPreclinicalFXIaBCL-2i
CapifutibatinibIncytePhase 3PCSK9BCL-2i
NBI-408NeurocrinePhase 2/3KRASG12DBCL-2i
HAL-996HalozymePhase 1/2BCL-2BCL-2i