← Pipeline|Zenozasiran

Zenozasiran

Preclinical
CIP-4431
Source: Trial-derived·Trials: 2
Modality
Cell Therapy
MOA
ALKi
Target
BET
Pathway
Proteasome
PsAFSGSNB
Development Pipeline
Preclinical
May 2023
Feb 2027
PreclinicalCurrent
NCT08519644
287 pts·FSGS
2024-072027-02·Not yet recruiting
NCT05782308
2,315 pts·NB
2023-05TBD·Recruiting
2,602 total pts2 indications
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2027-02-1310mo awayInterim· FSGS
Trial Timeline
Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027
Preclinical
Recruit…
Preclinical
Not yet…
Catalysts
Interim
2027-02-13 · 10mo away
FSGS
RecruitingNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT08519644PreclinicalFSGSNot yet recr...2876MWD
NCT05782308PreclinicalNBRecruiting2315VA
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-5767PfizerPhase 1/2BETCDK4/6i
MiriosocimabPfizerPhase 1PARPALKi
RHH-1969RocheApprovedBETCDK4/6i
NVS-5439NovartisPreclinicalBETAnti-Tau
MRK-7739Merck & CoPreclinicalIL-23ALKi
IvocapivasertibBristol-Myers SquibbPhase 1BETCDK4/6i
BMY-2495Bristol-Myers SquibbPhase 3KRASG12DALKi
DSN-5254Daiichi SankyoPhase 1B7-H3ALKi
SovacapivasertibAmgenPhase 3WEE1ALKi
ZanuratamabGilead SciencesPhase 1/2CDK2ALKi