← Pipeline|Tezetapinarof

Tezetapinarof

Phase 3
CGO-6895
Source: Trial-derived·Trials: 4
Modality
Nanobody
MOA
EZH2i
Target
VEGF
Pathway
mTOR
FTD
Development Pipeline
Preclinical
~Nov 2013
~Feb 2015
Phase 1
~May 2015
~Aug 2016
Phase 2
~Nov 2016
~Feb 2018
Phase 3
May 2018
Feb 2030
Phase 3Current
NCT08930071
2,613 pts·FTD
2022-112030-02·Recruiting
NCT06009027
1,922 pts·FTD
2024-042025-12·Not yet recruiting
NCT07377268
2,391 pts·FTD
2018-052029-01·Not yet recruiting
+1 more trial
7,966 total pts1 indication
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (4)
2025-12-223mo agoPh3 Readout· FTD
2028-10-072.5y awayPh3 Readout· FTD
2029-01-042.8y awayPh3 Readout· FTD
2030-02-133.9y awayPh3 Readout· FTD
Trial Timeline
Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
P3
Not yet…
P3
Recruit…
P3
Not yet…
P3
Active
Catalysts
Ph3 Readout
2025-12-22 · 3mo ago
FTD
Ph3 Readout
2028-10-07 · 2.5y away
FTD
Ph3 Readout
2029-01-04 · 2.8y away
FTD
Ph3 Readout
2030-02-13 · 3.9y away
FTD
RecruitingActiveNot yet recruiting|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT08930071Phase 3FTDRecruiting2613DAS28
NCT06009027Phase 3FTDNot yet recr...1922ORR
NCT07377268Phase 3FTDNot yet recr...2391SRI-4
NCT04653078Phase 3FTDActive1040DOR
Competitors (10)
DrugCompanyPhaseTargetMOA
ZanuderotideNovartisPhase 1/2VEGFCD3xCD20
AdagrazumabNovartisPhase 2/3Cl18.2EZH2i
RibotuximabMerck & CoPhase 2GPRC5DEZH2i
NVO-9615Novo NordiskPhase 2/3PRMT5EZH2i
TAK-8730TakedaPhase 2VEGFFXIai
GIL-2011Gilead SciencesPreclinicalVEGFSOS1i
BemazumabRegeneronPhase 1VEGFTROP-2 ADC
PemicapivasertibLegend BiotechPhase 3VEGFCDK4/6i
SematapinarofLegend BiotechNDA/BLAVEGFCGRPant
LEG-6533Legend BiotechNDA/BLAVEGFPARPi