← Pipeline|Tixatapinarof

Tixatapinarof

Phase 1/2
ARV-4994
Source: Trial-derived·Trials: 1
Modality
Cell Therapy
MOA
DLL3 ADC
Target
CDK2
Pathway
Angiogenesis
CSU
Development Pipeline
Preclinical
~May 2018
~Aug 2019
Phase 1
Nov 2019
Nov 2026
Phase 1Current
NCT03568461
2,508 pts·CSU
2019-112026-11·Not yet recruiting
2,508 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-11-228mo awayPh2 Data· CSU
Trial Timeline
Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q4
P1/2
Not yet…
Catalysts
Ph2 Data
2026-11-22 · 8mo away
CSU
Not yet recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT03568461Phase 1/2CSUNot yet recr...2508Safety
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-3703PfizerPhase 1/2CDK2CDK2i
NVS-3297NovartisPreclinicalCDK2MALT1i
NVS-4076NovartisPreclinicalTROP-2DLL3 ADC
RimamavacamtenMerck & CoPhase 1PI3KαDLL3 ADC
FixainavolisibTakedaPreclinicalCDK2IL-17i
AMG-1919AmgenPhase 2/3CDK2IL-13i
AMG-9654AmgenPhase 2GPRC5DDLL3 ADC
AMG-415AmgenPhase 1CDK2MDM2i
AMG-9052AmgenPhase 2/3CDK2USP1i
ZanuratamabGilead SciencesPhase 1/2CDK2ALKi