← Pipeline|Tezevorutinib

Tezevorutinib

Preclinical
ZEN-2806
Source: Trial-derived·Trials: 1
Modality
Vaccine
MOA
BTKi
Target
GPRC5D
Pathway
Checkpoint
FSGS
Development Pipeline
Preclinical
Jan 2017
Mar 2025
PreclinicalCurrent
NCT04475173
1,716 pts·FSGS
2017-012025-03·Active
1,716 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2025-03-041.1y agoInterim· FSGS
Trial Timeline
2017Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2
Preclinical
Active
Catalysts
Interim
2025-03-04 · 1.1y ago
FSGS
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04475173PreclinicalFSGSActive1716Biomarker
Competitors (10)
DrugCompanyPhaseTargetMOA
PexatenlimabNovartisPhase 1/2GPRC5DKIF18Ai
RibotuximabMerck & CoPhase 2GPRC5DEZH2i
AZN-8281AstraZenecaPhase 1SHP2BTKi
BMY-3371Bristol-Myers SquibbPhase 3WRNBTKi
BMY-9931Bristol-Myers SquibbPhase 1GPRC5DFXIai
NVO-7872Novo NordiskNDA/BLAB7-H3BTKi
NVO-7877Novo NordiskPreclinicalGPRC5DFXIai
NVO-6275Novo NordiskPhase 1SMN2BTKi
ZanumavacamtenGSKPhase 2/3TROP-2BTKi
TAK-2403TakedaPhase 2WEE1BTKi