← Pipeline|Terazanubrutinib

Terazanubrutinib

Phase 3
NBT-4735
Source: Trial-derived·Trials: 1
Modality
Gene Editing
MOA
ALKi
Target
KRASG12C
Pathway
Proteasome
PSPET
Development Pipeline
Preclinical
~Oct 2015
~Jan 2017
Phase 1
~Apr 2017
~Jul 2018
Phase 2
~Oct 2018
~Jan 2020
Phase 3
Apr 2020
Jun 2025
Phase 3Current
NCT07967485
586 pts·ET
2020-042025-06·Not yet recruiting
586 total pts1 indication
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2025-06-169mo agoPh3 Readout· ET
Trial Timeline
Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3
P3
Not yet…
Catalysts
Ph3 Readout
2025-06-16 · 9mo ago
ET
Not yet recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT07967485Phase 3ETNot yet recr...586ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
MiriosocimabPfizerPhase 1PARPALKi
JNJ-179Johnson & JohnsonApprovedKRASG12CBETi
MRK-7739Merck & CoPreclinicalIL-23ALKi
BMY-2495Bristol-Myers SquibbPhase 3KRASG12DALKi
BMY-4586Bristol-Myers SquibbPreclinicalKRASG12CIL-13i
DoxarapivirBristol-Myers SquibbPhase 3KRASG12CSOS1i
DSN-5254Daiichi SankyoPhase 1B7-H3ALKi
SovacapivasertibAmgenPhase 3WEE1ALKi
AMG-4531AmgenPhase 2/3KRASG12CPRMT5i
ZanuratamabGilead SciencesPhase 1/2CDK2ALKi