← Pipeline|Tezecapivasertib

Tezecapivasertib

Phase 2
DAR-5593
Source: Trial-derived·Trials: 2
Modality
mAb
MOA
FXIai
Target
Nectin-4
Pathway
Tau
Ewing Sarcoma
Development Pipeline
Preclinical
~Apr 2014
~Jul 2015
Phase 1
~Oct 2015
~Jan 2017
Phase 2
Apr 2017
Aug 2030
Phase 2Current
NCT06385724
1,807 pts·Ewing Sarcoma
2017-042025-09·Terminated
NCT04974355
2,447 pts·Ewing Sarcoma
2023-012030-08·Completed
4,254 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-09-137mo agoPh2 Data· Ewing Sarcoma
2030-08-134.4y awayPh2 Data· Ewing Sarcoma
Trial Timeline
2017Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
P2
Termina…
P2
Complet…
Catalysts
Ph2 Data
2025-09-13 · 7mo ago
Ewing Sarcoma
Ph2 Data
2030-08-13 · 4.4y away
Ewing Sarcoma
CompletedTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06385724Phase 2Ewing SarcomaTerminated1807OS
NCT04974355Phase 2Ewing SarcomaCompleted2447DOR
Competitors (10)
DrugCompanyPhaseTargetMOA
NVS-6360NovartisApprovedCD38FXIai
MRK-3745Merck & CoPhase 2WRNFXIai
MRK-2473Merck & CoPhase 1/2Nectin-4TYK2i
AZN-1715AstraZenecaPhase 3AHRFXIai
BMY-9931Bristol-Myers SquibbPhase 1GPRC5DFXIai
NVO-7877Novo NordiskPreclinicalGPRC5DFXIai
TAK-8730TakedaPhase 2VEGFFXIai
DSN-1421Daiichi SankyoPhase 3Nectin-4STINGag
SemazasiranBeiGenePhase 1PD-1FXIai
ION-3857IonisPreclinicalNectin-4TYK2i