← Pipeline|Elratapinarof

Elratapinarof

Preclinical
MAP-3327
Source: Trial-derived·Trials: 2
Modality
Radioligand
MOA
JAK1i
Target
Nectin-4
Pathway
T-cell
Gastric Ca
Development Pipeline
Preclinical
Jan 2017
Jan 2030
PreclinicalCurrent
NCT08117761
2,636 pts·Gastric Ca
2017-012030-01·Not yet recruiting
NCT08196959
1,750 pts·Gastric Ca
2022-07TBD·Active
4,386 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-07-049mo agoConference· Gastric Ca
2030-01-153.8y awayInterim· Gastric Ca
Trial Timeline
2017Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
Preclinical
Not yet…
Preclinical
Active
Catalysts
Conference
2025-07-04 · 9mo ago
Gastric Ca
Interim
2030-01-15 · 3.8y away
Gastric Ca
ActiveNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT08117761PreclinicalGastric CaNot yet recr...2636FEV1
NCT08196959PreclinicalGastric CaActive1750EDSS
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-7458Johnson & JohnsonPhase 1/2PD-1JAK1i
MRK-2473Merck & CoPhase 1/2Nectin-4TYK2i
GeliderotideSanofiPhase 1/2PRMT5JAK1i
PexaosocimabDaiichi SankyoPhase 2PD-1JAK1i
DSN-1421Daiichi SankyoPhase 3Nectin-4STINGag
AdagratapinarofVertex PharmaPreclinicalBCMAJAK1i
ARG-1924ArgenxPreclinicalDLL3JAK1i
ION-3857IonisPreclinicalNectin-4TYK2i
SemasacituzumabIlluminaPhase 3Nectin-4HPK1i
ROI-1081Roivant SciencesPhase 1/2PI3KαJAK1i