← Pipeline|Doxazasiran

Doxazasiran

Preclinical
PRI-4571
Source: Trial-derived·Trials: 2
Modality
Peptide
MOA
JAK1i
Target
KRASG12D
Pathway
T-cell
RB
Development Pipeline
Preclinical
Mar 2021
Dec 2030
PreclinicalCurrent
NCT07114075
2,069 pts·RB
2021-032030-12·Completed
NCT04673475
90 pts·RB
2025-102030-02·Not yet recruiting
2,159 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2030-02-193.9y awayInterim· RB
2030-12-244.7y awayInterim· RB
Trial Timeline
2021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
Preclinical
Complet…
Preclinical
Not yet…
Catalysts
Interim
2030-02-19 · 3.9y away
RB
Interim
2030-12-24 · 4.7y away
RB
CompletedNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07114075PreclinicalRBCompleted2069BodyWt
NCT04673475PreclinicalRBNot yet recr...90HbA1c
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-7458Johnson & JohnsonPhase 1/2PD-1JAK1i
RilulemzoparlimabNovartisPhase 2/3KRASG12DPD-L1i
BMY-2495Bristol-Myers SquibbPhase 3KRASG12DALKi
GeliderotideSanofiPhase 1/2PRMT5JAK1i
SNY-2934SanofiPhase 3KRASG12DUSP1i
TalainavolisibNovo NordiskPreclinicalKRASG12DPRMT5i
PexaosocimabDaiichi SankyoPhase 2PD-1JAK1i
GIL-2037Gilead SciencesApprovedKRASG12DMDM2i
AdagratapinarofVertex PharmaPreclinicalBCMAJAK1i
ARG-1924ArgenxPreclinicalDLL3JAK1i