← Pipeline|Capitapinarof

Capitapinarof

Preclinical
GAL-2731
Source: Trial-derived·Trials: 2
Modality
ADC
MOA
ALKi
Target
KIF18A
Pathway
Apoptosis
Cholangiocarcinoma
Development Pipeline
Preclinical
May 2024
Sep 2027
PreclinicalCurrent
NCT06449016
1,124 pts·Cholangiocarcinoma
2024-052027-09·Recruiting
NCT08884888
517 pts·Cholangiocarcinoma
2025-102027-09·Completed
1,641 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2027-09-111.4y awayInterim· Cholangiocarcinoma
2027-09-231.5y awayInterim· Cholangiocarcinoma
Trial Timeline
Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q4
Preclinical
Recruit…
Preclinical
Complet…
Catalysts
Interim
2027-09-11 · 1.4y away
Cholangiocarcinoma
Interim
2027-09-23 · 1.5y away
Cholangiocarcinoma
RecruitingCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06449016PreclinicalCholangiocarcinomaRecruiting1124PASI75
NCT08884888PreclinicalCholangiocarcinomaCompleted517eGFR
Competitors (10)
DrugCompanyPhaseTargetMOA
MiriosocimabPfizerPhase 1PARPALKi
NiranesiranJohnson & JohnsonPhase 2KIF18AEGFRi
MRK-7739Merck & CoPreclinicalIL-23ALKi
BMY-2495Bristol-Myers SquibbPhase 3KRASG12DALKi
DSN-5254Daiichi SankyoPhase 1B7-H3ALKi
SovacapivasertibAmgenPhase 3WEE1ALKi
ZanuratamabGilead SciencesPhase 1/2CDK2ALKi
GIL-2445Gilead SciencesPhase 2/3PSMAALKi
RiluinavolisibModernaNDA/BLAKIF18APLK4i
ALN-3284AlnylamPhase 2/3CDK2ALKi