← Pipeline|Elrarapivir

Elrarapivir

Phase 2
GUD-2445
Source: Trial-derived·Trials: 2
Modality
ASO
MOA
ALKi
Target
Nectin-4
Pathway
T-cell
NB
Development Pipeline
Preclinical
~Apr 2014
~Jul 2015
Phase 1
~Oct 2015
~Jan 2017
Phase 2
Apr 2017
Apr 2031
Phase 2Current
NCT06844499
2,659 pts·NB
2023-032031-04·Active
NCT08132899
1,472 pts·NB
2017-042028-07·Not yet recruiting
4,131 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-07-272.3y awayPh2 Data· NB
2031-04-245.1y awayPh2 Data· NB
Trial Timeline
2017Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3
P2
Not yet…
P2
Active
Catalysts
Ph2 Data
2028-07-27 · 2.3y away
NB
Ph2 Data
2031-04-24 · 5.1y away
NB
ActiveNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06844499Phase 2NBActive2659ACR20
NCT08132899Phase 2NBNot yet recr...1472Mayo
Competitors (10)
DrugCompanyPhaseTargetMOA
MiriosocimabPfizerPhase 1PARPALKi
MRK-7739Merck & CoPreclinicalIL-23ALKi
MRK-2473Merck & CoPhase 1/2Nectin-4TYK2i
BMY-2495Bristol-Myers SquibbPhase 3KRASG12DALKi
DSN-5254Daiichi SankyoPhase 1B7-H3ALKi
DSN-1421Daiichi SankyoPhase 3Nectin-4STINGag
SovacapivasertibAmgenPhase 3WEE1ALKi
ZanuratamabGilead SciencesPhase 1/2CDK2ALKi
GIL-2445Gilead SciencesPhase 2/3PSMAALKi
ALN-3284AlnylamPhase 2/3CDK2ALKi